CP-122,288

id: cp-122-288-254-10883104
title: CP-122,288
text: CP-122,288 is a drug which acts as a potent and selective agonist for the 5-HT1B, 5-HT1D and 5-HT1F serotonin receptor subtypes. It is a derivative of the migraine medication sumatriptan, but while CP-122,288 is 40,000 times more potent than sumatriptan as an inhibitor of neurogenic inflammation and plasma protein extravasation, it is only twice as potent as a constrictor of blood vessels. In human trials, CP-122,288 was not found to be effective as a treatment for migraine, but its selectivity
brand slug: wiki
category slug: encyclopedia
description: Chemical compound
original url: https://en.wikipedia.org/wiki/CP-122,288
date created:
date modified: 2024-01-13T11:06:26Z
main entity: {"identifier":"Q20707282","url":"https://www.wikidata.org/entity/Q20707282"}
image: {"content_url":"https://upload.wikimedia.org/wikipedia/commons/a/a9/CP-122%2C288_Structure.svg","width":6906,"height":3979}
fields total: 13
integrity: 15

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