WAY-161503

id: way-161503-281-16300799
title: WAY-161503
text: WAY-161503 is a full agonist of 5-HT2C receptors (Ki = 3.3 nM for displacement of DOI), ~6-fold less potent at 5-HT2A receptors (Ki = 18 nM) and 20-fold less potent at 5-HT2B receptors (Ki = 60 nM). In functional studies, it stimulates calcium mobilization coupled to 5-HT2C, 5-HT2B, and 5-HT2A receptors with EC50 values of 0.8, 1.8, and 7 nM, respectively. WAY-161503 has been reported to produce dose-dependent decreases in food intake in 24-hour fasted normal Sprague-Dawley rats, diet-induced ob
brand slug: wiki
category slug: encyclopedia
description: Chemical compound
original url: https://en.wikipedia.org/wiki/WAY-161503
date created:
date modified: 2022-11-08T19:31:47Z
main entity: {"identifier":"Q7946880","url":"https://www.wikidata.org/entity/Q7946880"}
image: {"content_url":"https://upload.wikimedia.org/wikipedia/commons/5/5c/WAY-161503.svg","width":512,"height":356}
fields total: 13
integrity: 15

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