LY-2459989
id:
ly-2459989-202-5791584
title:
LY-2459989
text:
LY-2459989 is a silent antagonist of the κ-opioid receptor (KOR) that has been developed by Eli Lilly as a radiotracer of that receptor, labeled either with carbon-11 or fluorine-18. It possesses high affinity for the KOR and is highly selective for it over the μ-opioid receptor and the δ-opioid receptor. LY-2459989 is a fluorine-containing analogue and follow-up compound of LY-2795050, the first KOR-selective antagonist radiotracer. Relative to LY-2795050, LY-2459989 displays 4-fold higher affi
brand slug:
wiki
category slug:
encyclopedia
description:
Chemical compound
original url:
https://en.wikipedia.org/wiki/LY-2459989
date created:
date modified:
2024-02-15T23:20:51Z
main entity:
{"identifier":"Q22906626","url":"https://www.wikidata.org/entity/Q22906626"}
image:
{"content_url":"https://upload.wikimedia.org/wikipedia/commons/4/4f/LY-2459989.svg","width":531,"height":297}
fields total:
13
integrity:
15