GSK-189254
id:
gsk-189254-317-10371294
title:
GSK-189254
text:
GSK-189,254 is a potent and selective H3 histamine receptor inverse agonist developed by GlaxoSmithKline. It has subnanomolar affinity for the H3 receptor (Ki = 0.2nM) and selectivity of over 10,000x for H3 over other histamine receptor subtypes. Animal studies have shown it to possess not only stimulant and nootropic effects, but also analgesic action suggesting a role for H3 receptors in pain processing in the spinal cord. GSK-189,254 and several other related drugs are currently being investi
brand slug:
wiki
category slug:
encyclopedia
description:
Chemical compound
original url:
https://en.wikipedia.org/wiki/GSK-189254
date created:
date modified:
2023-12-20T21:39:08Z
main entity:
{"identifier":"Q5514566","url":"https://www.wikidata.org/entity/Q5514566"}
image:
fields total:
13
integrity:
14