Desmethylclozapine

id: desmethylclozapine-248-7483064
title: Desmethylclozapine
text: N-Desmethylclozapine (NDMC), or norclozapine, is a major active metabolite of the atypical antipsychotic drug clozapine. Unlike clozapine, it possesses intrinsic activity at the D2/D3 receptors, and acts as a weak partial agonist at these sites similarly to aripiprazole and bifeprunox. Notably, NDMC has also been shown to act as a potent and efficacious agonist at the M1 and δ-opioid receptors, unlike clozapine as well. It was hypothesized that on account of these unique actions, NDMC might unde
brand slug: wiki
category slug: encyclopedia
description: Active metabolite of the drug clozapine
original url: https://en.wikipedia.org/wiki/Desmethylclozapine
date created:
date modified: 2023-10-28T23:54:24Z
main entity: {"identifier":"Q5264612","url":"https://www.wikidata.org/entity/Q5264612"}
image: {"content_url":"https://upload.wikimedia.org/wikipedia/commons/f/fd/Desmethylclozapine.svg","width":512,"height":478}
fields total: 13
integrity: 15

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