CI-966

id: ci-966-193-1930311
title: CI-966
text: CI-966 is a central nervous system depressant acting as a GABA reuptake inhibitor, specifically a highly potent and selective blocker of the GABA transporter 1 (GAT-1), and hence indirect and non-selective GABA receptor full agonist. It was investigated as a potential anticonvulsant, anxiolytic, and neuroprotective therapeutic but was discontinued during clinical development due to the incidence of severe adverse effects at higher doses and hence was never marketed. In a phase I human clinical t
brand slug: wiki
category slug: encyclopedia
description: Chemical compound
original url: https://en.wikipedia.org/wiki/CI-966
date created:
date modified: 2024-01-06T07:50:33Z
main entity: {"identifier":"Q15410874","url":"https://www.wikidata.org/entity/Q15410874"}
image: {"content_url":"https://upload.wikimedia.org/wikipedia/commons/2/2f/CI-966.svg","width":512,"height":384}
fields total: 13
integrity: 15

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