CGS-15943
id:
cgs-15943-196-11644626
title:
CGS-15943
text:
CGS-15943 is a drug which acts as a potent and reasonably selective antagonist for the adenosine receptors A1 and A2A, having a Ki of 3.3nM at A2A and 21nM at A1. It was one of the first adenosine receptor antagonists discovered that is not a xanthine derivative, instead being a triazoloquinazoline. Consequently, CGS-15943 has the advantage over most xanthine derivatives that it is not a phosphodiesterase inhibitor, and so has more a specific pharmacological effects profile. It produces similar
brand slug:
wiki
category slug:
encyclopedia
description:
Chemical compound
original url:
https://en.wikipedia.org/wiki/CGS-15943
date created:
date modified:
2022-10-28T14:39:56Z
main entity:
{"identifier":"Q5010994","url":"https://www.wikidata.org/entity/Q5010994"}
image:
{"content_url":"https://upload.wikimedia.org/wikipedia/commons/1/1b/CGS-15943_Structure.svg","width":5173,"height":4475}
fields total:
13
integrity:
15